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1991-1995
1. Theodorakis, E. A.; Royer, J.; Husson, H. P. "Asymmetric Synthesis XXIII. A 100% Cis Diastereoselectivity in the Synthesis of Enantiomerically Pure 2,6-Dialkylpiperidines". Synth. Commun. 1991, 21, 521-529. PDF File
2. Barton, D. H. R.; Jaszberenyi, J. Cs.; Theodorakis,
E. A. "O-Sulfinylation with Methanesulfonyl Cyanide or p-Toluenesulfonyl
Cyanide and DBU". Tetrahedron Lett. 1991,
32, 2585-2588.
PDF File
3. Barton, D. H. R.; Jaszberenyi, J. Cs.; Theodorakis, E. A. "Radical Nitrile Transfer with Methanesulfonyl Cyanide or p-Toluenesulfonyl Cyanide to Carbon Radicals Generated from the Acyl Derivatives of N-Hydroxy-2-Thiopyridone". Tetrahedron Lett. 1991, 32, 3321-3324. PDF File
4. Barton, D. H. R.; Jaszberenyi, J. Cs.; Theodorakis,
E. A. "O-Sulfinylation of Alcohols with Methanesulfonyl Cyanide or
p-Toluenesulfonyl Cyanide". Tetrahedron 1991,
47, 9167-9178.
PDF File
5. Barton, D. H. R.; Jaszberenyi, J. Cs.; Theodorakis, E. A. "The Invention of Radical Reactions. Part XXIII. New Reactions: Nitrile and Thiocyanate Transfer to Carbon Radicals from Sulfonyl Cyanides and Sulfonyl Isothiocyanates". Tetrahedron 1992, 47, 2613-2626. PDF File
6. Barton, D. H. R.; Jaszberenyi, J. Cs.; Theodorakis, E. A. "Nitrogen Transfer to Carbon Radicals". J. Am. Chem. Soc. 1992, 114, 5904-5905. PDF File
7. Barton, D. H. R.; Jaszberenyi, J. Cs.; Theodorakis, E. A.; Reibenspies, J. H. "The Invention of Radical Reactions. 30. Diazirines as Carbon Radical Traps. Mechanistic Aspects and Synthetic Applications of a Novel and Efficient Amination Process". J. Am. Chem. Soc. 1993, 115, 8050-8059. PDF File
8. Barton, D. H. R.; Parekh, S. I.; Tajbakhsh, M.; Theodorakis, E. A.; Tse, C.-L. "A Convenient and High Yielding Procedure for the Preparation of Isoselenocyanates. Synthesis and Reactivity of O-Alkylselenocarbamates". Tetrahedron 1994, 50, 639-654. PDF File
9. Nicolaou, K. C.; Pitsinos, E. N.; Theodorakis, E. A.; Saimoto, H.; Wrasidlo, W. "Synthetic Calicheamicin Mimics with Novel Initiation Mechanisms: DNA Cleavage, Cytotoxity and Apoptosis". Chemistry & Biology 1994, 1, 57-66. PDF File
10. Nicolaou, K. C.; Tiebes, J.; Theodorakis, E. A.; Rutjes, F. P. J. T.; Koide, K.; Sato, M.; Untersteller, E. "Total Synthesis of Truncated Brevetoxin B [AFGHIJK]". J. Am. Chem. Soc. 1994, 116, 9371-9372. PDF File
11. Nicolaou, K. C.; Theodorakis, E. A.; Rutjes, F.
P. J. T.; Tiebes, J.; Sato, M.; Untersteller, E.; Xiao, X.-Y. "Total
Synthesis of Brevetoxin B 1. CDEFG Framework". J. Am. Chem. Soc.
1995, 117, 1171-1172. PDF File
12. Nicolaou, K. C.; Rutjes, F. P. J. T.; Theodorakis,
E. A.; Tiebes, J.; Sato, M.; Untersteller, E. "Total Synthesis of
Brevetoxin B 2. Completion". J. Am. Chem. Soc. 1995,
117, 1173-1174.
PDF File
13. Nicolaou, K. C.; Hwang, C.-K.; Duggan, M. E.; Nugiel,
D. A.; Abe, Y.; Reddy, K. B.; DeFrees, S. A.; Reddy, D. R.; Awartani,
R. A.; Conley, S. R.; Rutjes, F. P. J. T.; Theodorakis, E. A. "Total
Synthesis of Brevetoxin B 1. First Generation Strategies and New Approaches
to Oxepane Systems". J. Am. Chem. Soc. 1995,
117, 10227-10238.
PDF File
14. Nicolaou, K. C.; Theodorakis, E. A.; Rutjes, F. P. J. T.; Sato, M.; Tiebes, J.; Xiao, X.-Y.; Hwang, C.-K.; Duggan, M. E.; Yang, Z; Couladouros, E. A.; Sato, F.; Shin, J.; He, H.-M.; Bleckman, T. "Total Synthesis of Brevetoxin B 2. Second Generation Strategies and Construction of the Dioxepane Region [DEFG]". J. Am. Chem. Soc. 1995, 117, 10239-10251. PDF File
15. Nicolaou, K. C.; Rutjes, F. P. J. T.; Theodorakis, E. A.; Tiebes, J.; Sato, M.; Untersteller, E. "Total Synthesis of Brevetoxin B 3. Final Strategy and Completion". J. Am. Chem. Soc. 1995, 117, 10252-10263. PDF File
16. Gawley, R. E.; Rein, K. S.; Jeglitsch, G.; Adams, D. J.; Theodorakis, E. A.; Tiebes, J.; Nicolaou, K. C.; Baden, D. G. "The Relationship of Brevetoxin "Length" and A-Ring Functionality to Binding and Activity in Neuronal Sodium Channels". Chemistry & Biology 1995, 2, 533-541. PDF File
17. Nicolaou, K. C.; Sato, M.; Theodorakis, E. A.; Miller, N. D. "Conversion of Thionoesters and Thionolactones to Ethers. A General and Efficient Radical Desulfurization". J. Chem. Soc. Chem. Commun. 1995, 1583-1585. PDF File